SA-4503
 | |
| Names | |
|---|---|
| IUPAC name
1-[2-(3,4-Dimethoxyphenyl)ethyl]-4-(3-phenylpropyl)piperazine | |
| Identifiers | |
165377-43-5  165377-44-6 (dihydrochloride)  | |
| 3D model (Jmol) | Interactive image |
| PubChem | 9954941 |
| |
| Properties | |
| C23H32N2O2 | |
| Molar mass | 368.52 g·mol−1 |
| Except where otherwise noted, data are given for materials in their standard state (at 25 °C [77 °F], 100 kPa). | |
| verify (what is ?) | |
| Infobox references | |
SA 4503 is a sigma receptor agonist.[1][2][3]
References
- ↑ Matsuno K, Nakazawa M, Okamoto K, Kawashima Y, Mita S (1996). "Binding properties of SA4503, a novel and selective sigma 1 receptor agonist". European Journal of Pharmacology. 306 (1-3): 271–9. doi:10.1016/0014-2999(96)00201-4. PMID 8813641.
- ↑ Skuza G, Rogóz Z (2006). "The synergistic effect of selective sigma receptor agonists and uncompetitive NMDA receptor antagonists in the forced swim test in rats". J. Physiol. Pharmacol. 57 (2): 217–29. PMID 16845227.
- ↑ Xu R, Lord SA, Peterson RM, Fergason-Cantrell EA, Lever JR, Lever SZ (January 2015). "Ether modifications to 1-[2-(3,4-dimethoxyphenyl)ethyl]-4-(3-phenylpropyl)piperazine (SA4503): effects on binding affinity and selectivity for sigma receptors and monoamine transporters.". Bioorganic & Medicinal Chemistry. 23 (1): 222–230. doi:10.1016/j.bmc.2014.11.007.
External links
- SA 4503 at the US National Library of Medicine Medical Subject Headings (MeSH)
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